ABSTRACT
Instant Notes in Medicinal Chemistry provides concise coverage for undergraduates studying medicinal chemistry as part of a science, pharmacy or medical course. It is a truly multidisciplinary subject involving such subject specialities as organic chemistry, pharmacology, biochemistry, physiology, microbiology, toxicology, genetics and computer mod
TABLE OF CONTENTS
section Section A|1 pages
The science of medicinal chemistry
section Section B|1 pages
Drug targets
section Section C|1 pages
Pharmacokinetics
section Section D|1 pages
Biological testing and bioassays
section Section E|1 pages
Drug discovery
section Section F|1 pages
Synthesis
section Section G|1 pages
Structure–activity relationships
section Section H|1 pages
Target orientated drug design
section Section I|1 pages
Pharmacokinetic orientated drug design
section Section J|1 pages
Patenting and Manufacture
section Section K|1 pages
Preclinical testing and clinical trials
section Section L|1 pages
Case study: inhibitors of EGF-receptor kinase
section Section M|1 pages
History of medicinal chemistry